Các bài viết có thể truy cập công khai - Peter ScammellsTìm hiểu thêm
Không có ở bất kỳ nơi nào: 27
Biased agonism at G protein‐coupled receptors: the promise and the challenges—a medicinal chemistry perspective
J Shonberg, L Lopez, PJ Scammells, A Christopoulos, B Capuano, ...
Medicinal research reviews 34 (6), 1286-1330, 2014
Các cơ quan ủy nhiệm: Australian Research Council, National Health and Medical Research Council …
A structure–activity analysis of biased agonism at the dopamine D2 receptor
J Shonberg, CK Herenbrink, L Lopez, A Christopoulos, PJ Scammells, ...
Journal of medicinal chemistry 56 (22), 9199-9221, 2013
Các cơ quan ủy nhiệm: Australian Research Council, National Health and Medical Research Council …
The hybrid molecule, VCP746, is a potent adenosine A2B receptor agonist that stimulates anti-fibrotic signalling
EA Vecchio, CH Chuo, JA Baltos, L Ford, PJ Scammells, BH Wang, ...
Biochemical pharmacology 117, 46-56, 2016
Các cơ quan ủy nhiệm: Australian Research Council, National Health and Medical Research Council …
Ligand-Induced Conformational Change of Plasmodium falciparum AMA1 Detected Using 19F NMR
X Ge, CA MacRaild, SM Devine, CO Debono, G Wang, PJ Scammells, ...
Journal of Medicinal Chemistry 57 (15), 6419-6427, 2014
Các cơ quan ủy nhiệm: National Health and Medical Research Council, Australia
The synthesis and biological evaluation of multifunctionalised derivatives of noscapine as cytotoxic agents
AJ DeBono, SJ Mistry, J Xie, D Muthiah, J Phillips, S Ventura, ...
ChemMedChem 9 (2), 399-410, 2014
Các cơ quan ủy nhiệm: Australian Research Council
Synthesis and pharmacological evaluation of analogues of benzyl quinolone carboxylic acid (BQCA) designed to bind irreversibly to an allosteric site of the M1 muscarinic …
BJ Davie, C Valant, JM White, PM Sexton, B Capuano, A Christopoulos, ...
Journal of medicinal chemistry 57 (12), 5405-5418, 2014
Các cơ quan ủy nhiệm: Australian Research Council, National Health and Medical Research Council …
Hydroxamic Acid Inhibitors Provide Cross-Species Inhibition of Plasmodium M1 and M17 Aminopeptidases
NB Vinh, N Drinkwater, TR Malcolm, M Kassiou, L Lucantoni, PM Grin, ...
Journal of medicinal chemistry 62 (2), 622-640, 2018
Các cơ quan ủy nhiệm: National Health and Medical Research Council, Australia, Canadian Institutes …
Rapid Elaboration of Fragments into Leads by X-ray Crystallographic Screening of Parallel Chemical Libraries (REFiLX)
MR Bentley, OV Ilyichova, G Wang, ML Williams, G Sharma, WS Alwan, ...
Journal of Medicinal Chemistry 63 (13), 6863-6875, 2020
Các cơ quan ủy nhiệm: National Health and Medical Research Council, Australia
Novel human aminopeptidase N inhibitors: Discovery and optimization of subsite binding interactions
J Lee, NB Vinh, N Drinkwater, W Yang, K Kannan Sivaraman, ...
Journal of Medicinal Chemistry 62 (15), 7185-7209, 2019
Các cơ quan ủy nhiệm: National Health and Medical Research Council, Australia
VCP746, a novel A1 adenosine receptor biased agonist, reduces hypertrophy in a rat neonatal cardiac myocyte model
CH Chuo, SM Devine, PJ Scammells, H Krum, A Christopoulos, LT May, ...
Clinical and Experimental Pharmacology and Physiology 43 (10), 976-982, 2016
Các cơ quan ủy nhiệm: Australian Research Council, National Health and Medical Research Council …
Discovery and development of 2-aminobenzimidazoles as potent antimalarials
SM Devine, MP Challis, JK Kigotho, G Siddiqui, A De Paoli, CA MacRaild, ...
European Journal of Medicinal Chemistry 221, 113518, 2021
Các cơ quan ủy nhiệm: National Health and Medical Research Council, Australia
Synthesis and Pharmacological Evaluation of Heterocyclic Carboxamides: Positive Allosteric Modulators of the M1 Muscarinic Acetylcholine Receptor with Weak …
JCC Dallagnol, E Khajehali, ET Van Der Westhuizen, M Jörg, C Valant, ...
Journal of Medicinal Chemistry 61 (7), 2875-2894, 2018
Các cơ quan ủy nhiệm: Australian Research Council, National Health and Medical Research Council …
Overcoming P-glycoprotein–mediated drug resistance with noscapine derivatives
D Muthiah, GK Henshaw, AJ DeBono, B Capuano, PJ Scammells, ...
Drug Metabolism and Disposition 47 (2), 164-172, 2019
Các cơ quan ủy nhiệm: Worldwide Cancer Research, UK
Subtle Modifications to the Indole-2-carboxamide Motif of the Negative Allosteric Modulator N-((trans)-4-(2-(7-Cyano-3, 4-dihydroisoquinolin-2 (1 H)-yl) ethyl) cyclohexyl)-1 H …
A Kopinathan, C Draper-Joyce, M Szabo, A Christopoulos, PJ Scammells, ...
Journal of Medicinal Chemistry 62 (1), 371-377, 2018
Các cơ quan ủy nhiệm: National Health and Medical Research Council, Australia
Structure and substrate fingerprint of aminopeptidase P from Plasmodium falciparum
N Drinkwater, KK Sivaraman, RS Bamert, W Rut, K Mohamed, NB Vinh, ...
Biochemical Journal 473 (19), 3189-3204, 2016
Các cơ quan ủy nhiệm: National Health and Medical Research Council, Australia
Utility of iron nanoparticles and a solution-phase iron species for the N-demethylation of alkaloids
JK Awalt, R Lam, B Kellam, B Graham, PJ Scammells, RD Singer
Green Chemistry 19 (11), 2587-2594, 2017
Các cơ quan ủy nhiệm: Natural Sciences and Engineering Research Council of Canada
Development of a Photoactivatable Allosteric Ligand for the M1 Muscarinic Acetylcholine Receptor
BJ Davie, PM Sexton, B Capuano, A Christopoulos, PJ Scammells
ACS chemical neuroscience 5 (10), 902-907, 2014
Các cơ quan ủy nhiệm: Australian Research Council, National Health and Medical Research Council …
Solution NMR characterization of apical membrane antigen 1 and small molecule interactions as a basis for designing new antimalarials
B Krishnarjuna, SS Lim, SM Devine, CO Debono, R Lam, ...
Journal of Molecular Recognition 29 (6), 281-291, 2016
Các cơ quan ủy nhiệm: National Health and Medical Research Council, Australia, Department of …
Diffusion tensor imaging evaluation of axonal/white matter remodeling in a mouse model of diabetic stroke treated with novel p38 MAPK inhibitor, VCP979
Y Cai, C Lu, T Xu, Y Ma, S Min, P Scammells, B Wang, S Ju
Journal of Biomedical Nanotechnology 14 (3), 585-593, 2018
Các cơ quan ủy nhiệm: National Health and Medical Research Council, Australia, National Natural …
Effect of Linker Length and Composition on Heterobivalent Ligand‐Mediated Receptor Cross‐Talk between the A1 Adenosine and β2 Adrenergic Receptors
N Barlow, SP Baker, PJ Scammells
ChemMedChem 8 (12), 2036-2046, 2013
Các cơ quan ủy nhiệm: Australian Research Council
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