Radiosynthesis and in vivo evaluation of a series of substituted 11C-phenethylamines as 5-HT2A agonist PET tracers A Ettrup, M Hansen, MA Santini, J Paine, N Gillings, M Palner, S Lehel, ... European journal of nuclear medicine and molecular imaging 38, 681-693, 2011 | 137 | 2011 |
Synthesis and Structure–Activity Relationships of N-Benzyl Phenethylamines as 5-HT2A/2C Agonists M Hansen, K Phonekeo, JS Paine, S Leth-Petersen, M Begtrup, ... ACS chemical neuroscience 5 (3), 243-249, 2014 | 132 | 2014 |
Serotonin 2A Receptor Agonist Binding in the Human Brain with [11C]Cimbi-36 A Ettrup, S da Cunha-Bang, B McMahon, S Lehel, A Dyssegaard, ... Journal of Cerebral Blood Flow & Metabolism 34 (7), 1188-1196, 2014 | 111 | 2014 |
Characterization of [11C] Cimbi-36 as an agonist PET radioligand for the 5-HT2A and 5-HT2C receptors in the nonhuman primate brain SJ Finnema, V Stepanov, A Ettrup, R Nakao, N Amini, M Svedberg, ... Neuroimage 84, 342-353, 2014 | 73 | 2014 |
Mechanistic Study of the sPLA2-Mediated Hydrolysis of a Thio-ester Pro Anticancer Ether Lipid L Linderoth, P Fristrup, M Hansen, F Melander, R Madsen, TL Andresen, ... Journal of the American Chemical Society 131 (34), 12193-12200, 2009 | 71 | 2009 |
Radiosynthesis and evaluation of 11C-CIMBI-5 as a 5-HT2A receptor agonist radioligand for PET A Ettrup, M Palner, N Gillings, MA Santini, M Hansen, BR Kornum, ... Journal of Nuclear Medicine 51 (11), 1763-1770, 2010 | 60 | 2010 |
Extensive Rigid Analogue Design Maps the Binding Conformation of Potent N-Benzylphenethylamine 5-HT2A Serotonin Receptor Agonist Ligands JI Juncosa Jr, M Hansen, LA Bonner, JP Cueva, R Maglathlin, ... ACS chemical neuroscience 4 (1), 96-109, 2013 | 59 | 2013 |
Hallucinogen-like effects of 2-([2-(4-cyano-2,5-dimethoxyphenyl) ethylamino]methyl)phenol (25CN-NBOH), a novel N-benzylphenethylamine with 100-fold selectivity for 5-HT … WE Fantegrossi, BW Gray, JM Bailey, DA Smith, M Hansen, JL Kristensen Psychopharmacology 232, 1039-1047, 2015 | 56 | 2015 |
Preclinical Safety Assessment of the 5-HT2A Receptor Agonist PET Radioligand [11C]Cimbi-36 A Ettrup, S Holm, M Hansen, M Wasim, MA Santini, M Palner, J Madsen, ... Molecular imaging and biology 15, 376-383, 2013 | 49 | 2013 |
Palladium‐Catalyzed C H Activation of N‐Allyl Imines: Regioselective Allylic Alkylations to Deliver Substituted Aza‐1, 3‐Dienes BM Trost, S Mahapatra, M Hansen Angewandte Chemie International Edition 54 (20), 6032-6036, 2015 | 34 | 2015 |
Synthesis and pharmacological evaluation of N-benzyl substituted 4-bromo-2, 5-dimethoxyphenethylamines as 5-HT2A/2C partial agonists M Hansen, SE Jacobsen, S Plunkett, GE Liebscher, JD McCorvy, ... Bioorganic & medicinal chemistry 23 (14), 3933-3937, 2015 | 33 | 2015 |
Correlating the Metabolic Stability of Psychedelic 5-HT2A Agonists with Anecdotal Reports of Human Oral Bioavailability S Leth-Petersen, C Bundgaard, M Hansen, MA Carnerup, J Kehler, ... Neurochemical research 39, 2018-2023, 2014 | 31 | 2014 |
A prodrug approach involving in situ depot formation to achieve localized and sustained action of diclofenac after joint injection M Thing, L Ågårdh, S Larsen, R Rasmussen, J Pallesen, N Mertz, ... Journal of Pharmaceutical Sciences 103 (12), 4021-4029, 2014 | 14 | 2014 |
Synthesis of new diverse macrocycles from diol precursors CM Madsen, M Hansen, MV Thrane, MH Clausen Tetrahedron 66 (52), 9849-9859, 2010 | 13 | 2010 |
Accelerating preclinical PET-screening: reductive amination with [11 C] methoxybenzaldehydes MM Herth, S Leth-Petersen, S Lehel, M Hansen, GM Knudsen, N Gillings, ... RSC Advances 4 (41), 21347-21350, 2014 | 10 | 2014 |
Development of an F-18-labelled 5-HT2A receptor agonist PET radioligand A Ettrup, M Hansen, N Gillings, A Dyssegaard, S Lehel, HD Hansen, ... JOURNAL OF CEREBRAL BLOOD FLOW AND METABOLISM 32, S109-S109, 2012 | 4 | 2012 |
In vivo evaluation of a series of substituted C-11-phenetylamines as 5-HT2A agonist PET tracers A Ettrup, M Hansen, MA Santini, J Paine, N Gillings, M Palner, S Lehel, ... NeuroImage 52 (Suppl. 1), 2010 | 4 | 2010 |
New macrocycles from diversity-oriented synthesis CM Madsen, M Hansen, MV Thrane, MH Clausen ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY 238, 2009 | | 2009 |