Delayed functional expression of neuronal chemokine receptors following focal nerve demyelination in the rat: a mechanism for the development of chronic sensitization of … S Bhangoo, D Ren, RJ Miller, KJ Henry, J Lineswala, C Hamdouchi, B Li, ... Molecular pain 3, 1744-8069-3-38, 2007 | 208 | 2007 |
Lithium perchlorate catalyzed conjugate addition of O-silylated ketene acetals to hindered α, β-unsaturated carbonyl compounds at atmospheric pressure PA Grieco, RJ Cooke, KJ Henry, JM VanderRoest Tetrahedron letters 32 (36), 4665-4668, 1991 | 80 | 1991 |
Chelation controlled addition of allylstannanes to aldehydes in lithium perchlorate-diethyl ether KJ Henry Jr, PA Grieco, CT Jagoe Tetrahedron letters 33 (14), 1817-1820, 1992 | 78 | 1992 |
7-phenyl-isoquinoline-5-sulfonylamino derivatives as inhibitors of akt (protein kinase B) DA Barda, KJ Henry Jr, J Huang, S Joseph, HS Lin, ME Richett US Patent 7,449,477, 2008 | 70 | 2008 |
Cyclopropanation of glycals: Application to the synthesis of 2-deoxy-2-vinyl glycosides KJ Henry Jr, B Fraser-Reid Tetrahedron letters 36 (49), 8901-8904, 1995 | 51 | 1995 |
Free radical methodology for carbohydrate to carbocycle transformations: an efficient synthesis of the tricyclic dihydrofuran portion of azadirachtin KJ Henry Jr, B Fraser-Reid The Journal of Organic Chemistry 59 (18), 5128-5129, 1994 | 47 | 1994 |
Pyrrolidine-3-carboxylic Acids as Endothelin Antagonists. 3. Discovery of a Potent, 2-Nonaryl, Highly Selective ETA Antagonist (A-216546) G Liu, KJ Henry, BG Szczepankiewicz, M Winn, NS Kozmina, SA Boyd, ... Journal of medicinal chemistry 41 (17), 3261-3275, 1998 | 38 | 1998 |
Direct substitution of secondary allylic alcohols with O-silylated ketene acetals in 3.0 M lithium perchlorate-diethyl ether-An alternative to the [1, 3] sigmatropic … PA Grieco, JL Collins, KJ Henry Jr Tetrahedron letters 33 (33), 4735-4738, 1992 | 37 | 1992 |
Endothelin antagonists M Winn, SA Boyd, CW Hutchins, HS Jae, AS Tasker, TW Von Geldern, ... US Patent 6,162,927, 2000 | 35 | 2000 |
Discovery of a series of cyclohexylethylamine-containing protein farnesyltransferase inhibitors exhibiting potent cellular activity KJ Henry, J Wasicak, AS Tasker, J Cohen, P Ewing, M Mitten, JJ Larsen, ... Journal of medicinal chemistry 42 (23), 4844-4852, 1999 | 34 | 1999 |
Total synthesis of (±)-sesbanimide A and B PA Grieco, KJ Henry, JJ Nunes, JE Matt Journal of the Chemical Society, Chemical Communications, 368-370, 1992 | 29 | 1992 |
Discovery of a series of pyrrolidine-based endothelin receptor antagonists with enhanced ETA receptor selectivity SA Boyd, RA Mantei, AS Tasker, G Liu, BK Sorensen, KJ Henry Jr, ... Bioorganic & medicinal chemistry 7 (6), 991-1002, 1999 | 27 | 1999 |
Endothelin antagonists M Winn, SA Boyd, CW Hutchins, HS Jae, AS Tasker, TW Von Geldern, ... US Patent 6,946,481, 2005 | 26 | 2005 |
Inhibitors of protein isoprenyl transferases SM Sebti, AD Hamilton, DJ Augeri, KJ Barr, SA Fakhoury, DA Janowick, ... US Patent 6,310,095, 2001 | 25 | 2001 |
Potent inhibitors of protein farnesyltransferase: heteroarenes as cysteine replacements W Shen, S Fakhoury, G Donner, K Henry, J Lee, H Zhang, J Cohen, ... Bioorganic & medicinal chemistry letters 9 (5), 703-708, 1999 | 25 | 1999 |
3-(2-acylamino-1-hydroxyethyl)-morpholine derivatives and their use as BACE inhibitors HB Broughton, RD Dally, TB Durham, MR Gonzalez-Garcia, PJ Hahn, ... US Patent 7,745,438, 2010 | 24 | 2010 |
A novel approach to iboga alkaloids: Total synthesis of (±)-ibogamine and (±)-epi-ibogamine KJ Henry Jr, PA Grieco, WJ DuBay Tetrahedron letters 37 (46), 8289-8292, 1996 | 20 | 1996 |
Endothelin antagonists M Winn, SA Boyd, CW Hutchins, HS Jae, AS Tasker, TW Von Geldern, ... US Patent 7,208,517, 2007 | 18 | 2007 |
Inhibitors of protein isoprenyl transferases SM Sebti, AD Hamilton, KJ Barr, SA Fakhoury, SJ O'connor, ... US Patent 6,221,865, 2001 | 18 | 2001 |
AKT inhibitors DW Beight, TP Burkholder, JR Clayton, MJ Eggen, KJ Henry Jr, DM Johns, ... US Patent 8,436,002, 2013 | 16 | 2013 |