Članki z zahtevami za javni dostop - R. Kip GuyVeč o tem
Ni na voljo nikjer: 8
Quinolone-3-diarylethers: a new class of antimalarial drug
A Nilsen, AN LaCrue, KL White, IP Forquer, RM Cross, J Marfurt, ...
Science translational medicine 5 (177), 177ra37-177ra37, 2013
Zahteve: US National Institutes of Health
Safety, tolerability, pharmacokinetics, and antimalarial efficacy of a novel Plasmodium falciparum ATP4 inhibitor SJ733: a first-in-human and induced blood-stage malaria phase …
AH Gaur, JS McCarthy, JC Panetta, RH Dallas, J Woodford, L Tang, ...
The Lancet Infectious Diseases 20 (8), 964-975, 2020
Zahteve: National Health and Medical Research Council, Australia
Synthesis and Structure–Activity Relationship of Dual-Stage Antimalarial Pyrazolo[3,4-b]pyridines
S Eagon, JT Hammill, M Sigal, KJ Ahn, JE Tryhorn, G Koch, B Belanger, ...
Journal of Medicinal Chemistry 63 (20), 11902-11919, 2020
Zahteve: Wellcome Trust
LC-MS- and 1H NMR Spectroscopy-Guided Identification of Antifungal Diterpenoids from Sagittaria latifolia
RR Ravu, MR Jacob, C Jeffries, Y Tu, SI Khan, AK Agarwal, RK Guy, ...
Journal of Natural Products 78 (9), 2255-2259, 2015
Zahteve: US National Institutes of Health
Transition-metal-free one-pot tandem synthesis of 4-quinolone and 4H-thiochromen-4-one derivatives through sequential nucleophilic addition–elimination–SNAr reaction
D Wang, P Sun, P Jia, J Peng, Y Yue, C Chen
Synthesis 49 (18), 4309-4320, 2017
Zahteve: National Natural Science Foundation of China
Ligand competition binding assay for the androgen receptor
C Féau, LA Arnold, A Kosinski, RK Guy
Androgen Action: Methods and Protocols, 59-68, 2011
Zahteve: US National Institutes of Health
Current and emerging therapy for improving outcomes in patients with intraocular retinoblastoma
RC Brennan, EM Pritchard, RK Guy, MA Dyer, MW Wilson
Expert Opinion on Orphan Drugs 3 (10), 1155-1166, 2015
Zahteve: US National Institutes of Health
Pharmacological stabilization of ΔF508-CFTR at the cell surface: design of CAL-selective PDZ inhibitors
P Cushing, P Boisguérin, L Vouilleme, M Pellegrini, D Mierke, D Smithson, ...
Journal of Cystic Fibrosis 9, S15, 2010
Zahteve: US National Institutes of Health
Na voljo nekje: 102
Chemical genetics of Plasmodium falciparum
WA Guiguemde, AA Shelat, D Bouck, S Duffy, GJ Crowther, PH Davis, ...
Nature 465 (7296), 311-315, 2010
Zahteve: US National Institutes of Health, Howard Hughes Medical Institute
Open source drug discovery with the malaria box compound collection for neglected diseases and beyond
WC Van Voorhis, JH Adams, R Adelfio, V Ahyong, MH Akabas, P Alano, ...
PLoS pathogens 12 (7), e1005763, 2016
Zahteve: US National Science Foundation, Bill & Melinda Gates Foundation, US National …
(+)-SJ733, a clinical candidate for malaria that acts through ATP4 to induce rapid host-mediated clearance of Plasmodium
MB Jiménez-Díaz, D Ebert, Y Salinas, A Pradhan, AM Lehane, ...
Proceedings of the National Academy of Sciences 111 (50), E5455-E5462, 2014
Zahteve: US National Institutes of Health, Howard Hughes Medical Institute, National …
Identification and characterization of the first small molecule inhibitor of MDMX
D Reed, Y Shen, AA Shelat, LA Arnold, AM Ferreira, F Zhu, N Mills, ...
Journal of Biological Chemistry 285 (14), 10786-10796, 2010
Zahteve: US National Institutes of Health, Howard Hughes Medical Institute
Efficacy of retinoids in IKZF1-mutated BCR-ABL1 acute lymphoblastic leukemia
ML Churchman, J Low, C Qu, EM Paietta, LH Kasper, Y Chang, ...
Cancer cell 28 (3), 343-356, 2015
Zahteve: US National Institutes of Health
Targeting the binding function 3 (BF3) site of the human androgen receptor through virtual screening.
NA Lack, P Axerio-Cilies, P Tavassoli, FQ Han, KH Chan, C Feau, ...
Journal of medicinal chemistry 54 (24), 8563-8573, 2011
Zahteve: US National Institutes of Health, Canadian Institutes of Health Research
NALP3 inflammasome upregulation and CASP1 cleavage of the glucocorticoid receptor cause glucocorticoid resistance in leukemia cells
SW Paugh, EJ Bonten, D Savic, LB Ramsey, WE Thierfelder, P Gurung, ...
Nature genetics 47 (6), 607-614, 2015
Zahteve: US National Institutes of Health
Global phenotypic screening for antimalarials
WA Guiguemde, AA Shelat, JF Garcia-Bustos, TT Diagana, FJ Gamo, ...
Chemistry & biology 19 (1), 116-129, 2012
Zahteve: US National Institutes of Health
Targeting the regulation of androgen receptor signaling by the heat shock protein 90 cochaperone FKBP52 in prostate cancer cells
JT De Leon, A Iwai, C Feau, Y Garcia, HA Balsiger, CL Storer, RM Suro, ...
Proceedings of the National Academy of Sciences 108 (29), 11878-11883, 2011
Zahteve: US National Institutes of Health
Pemetrexed and gemcitabine as combination therapy for the treatment of Group3 medulloblastoma
M Morfouace, A Shelat, M Jacus, BB Freeman, D Turner, S Robinson, ...
Cancer cell 25 (4), 516-529, 2014
Zahteve: US National Institutes of Health, National Institute of Health and Medical …
An integrated in vitro and in vivo high-throughput screen identifies treatment leads for ependymoma
JM Atkinson, AA Shelat, AM Carcaboso, TA Kranenburg, LA Arnold, ...
Cancer cell 20 (3), 384-399, 2011
Zahteve: US National Institutes of Health
Non-competitive androgen receptor inhibition in vitro and in vivo
JO Jones, EC Bolton, Y Huang, C Feau, RK Guy, KR Yamamoto, B Hann, ...
Proceedings of the National Academy of Sciences 106 (17), 7233-7238, 2009
Zahteve: US National Institutes of Health
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