| Strategies to improve plasma half life time of peptide and protein drugs M Werle, A Bernkop-Schnürch Amino acids 30, 351-367, 2006 | 810 | 2006 |
| Natural and synthetic polymers as inhibitors of drug efflux pumps M Werle Pharmaceutical Research 25, 500-511, 2008 | 243 | 2008 |
| Glutathione and thiolated chitosan inhibit multidrug resistance P-glycoprotein activity in excised small intestine M Werle, M Hoffer Journal of controlled release 111 (1-2), 41-46, 2006 | 201 | 2006 |
| Synthesis and in vitro evaluation of thiolated hyaluronic acid for mucoadhesive drug delivery K Kafedjiiski, RKR Jetti, F Föger, H Hoyer, M Werle, M Hoffer, ... International journal of pharmaceutics 343 (1-2), 48-58, 2007 | 159 | 2007 |
| A mucoadhesive nanoparticulate system for the simultaneous delivery of macromolecules and permeation enhancers to the intestinal mucosa A Makhlof, M Werle, Y Tozuka, H Takeuchi Journal of controlled release 149 (1), 81-88, 2011 | 154 | 2011 |
| Modified chitosans for oral drug delivery M Werle, H Takeuchi, A Bernkop-Schnürch Journal of pharmaceutical sciences 98 (5), 1643-1656, 2009 | 150 | 2009 |
| Nanoparticles of glycol chitosan and its thiolated derivative significantly improved the pulmonary delivery of calcitonin A Makhlof, M Werle, Y Tozuka, H Takeuchi International journal of pharmaceutics 397 (1-2), 92-95, 2010 | 140 | 2010 |
| Chitosan–aprotinin coated liposomes for oral peptide delivery: Development, characterisation and in vivo evaluation M Werle, H Takeuchi International journal of pharmaceutics 370 (1-2), 26-32, 2009 | 139 | 2009 |
| Synthesis and in Vitro Evaluation of a Novel Chitosan–Glutathione Conjugate K Kafedjiiski, F Föger, M Werle, A Bernkop-Schnürch Pharmaceutical research 22, 1480-1488, 2005 | 132 | 2005 |
| The potential of cystine-knot microproteins as novel pharmacophoric scaffolds in oral peptide drug delivery M Werle, T Schmitz, HL Huang, A Wentzel, H Kolmar, ... Journal of drug targeting 14 (3), 137-146, 2006 | 115 | 2006 |
| Thiolated chitosans: useful excipients for oral drug delivery M Werle, A Bernkop‐Schnürch Journal of Pharmacy and Pharmacology 60 (3), 273-281, 2008 | 97 | 2008 |
| Improved synthesis and in vitro characterization of chitosan–thioethylamidine conjugate K Kafedjiiski, M Hoffer, M Werle, A Bernkop-Schnürch Biomaterials 27 (1), 127-135, 2006 | 79 | 2006 |
| Evaluation and improvement of the properties of the novel cystine-knot microprotein McoEeTI for oral administration M Werle, K Kafedjiiski, H Kolmar, A Bernkop-Schnürch International journal of pharmaceutics 332 (1-2), 72-79, 2007 | 70 | 2007 |
| Oral gene delivery: Strategies to improve stability of pDNA towards intestinal digestion B Loretz, F Föger, M Werle, A Bernkop-Schnuerch Journal of drug targeting 14 (5), 311-319, 2006 | 59 | 2006 |
| Carbopol-lectin conjugate coated liposomes for oral peptide delivery M Werle, A Makhlof, H Takeuchi Chemical and Pharmaceutical Bulletin 58 (3), 432-434, 2010 | 46 | 2010 |
| Oral protein delivery: a patent review of academic and industrial approaches M Werle, A Makhlof, H Takeuchi Recent patents on drug delivery & formulation 3 (2), 94-104, 2009 | 43 | 2009 |
| Degradation of teriparatide by gastro-intestinal proteolytic enzymes M Werle, A Samhaber, A Bernkop-Schnürch Journal of drug targeting 14 (3), 109-115, 2006 | 33 | 2006 |
| Design and evaluation of a chitosan–aprotinin conjugate for the peroral delivery of therapeutic peptides and proteins susceptible to enzymatic degradation M Werle, B Loretz, D Entstrasser, F Föger Journal of drug targeting 15 (5), 327-333, 2007 | 31 | 2007 |
| Effect of a thiolated polymer on oral paclitaxel absorption and tumor growth in rats F Föger, S Malaivijitnond, T Wannaprasert, C Huck, A Bernkop-Schnürch, ... Journal of drug targeting 16 (2), 149-155, 2008 | 29 | 2008 |
| Mucoadhesive drug carriers and polymers for effective drug delivery A Makhlof, M Werle, H Takeuchi Journal of drug delivery science and technology 18 (6), 375-386, 2008 | 28 | 2008 |