Optically active N-protected. alpha.-amino aldehydes in organic synthesis J Jurczak, A Golebiowski Chemical Reviews 89 (1), 149-164, 1989 | 624 | 1989 |
Enantioselective synthesis through enzymatic asymmetrization E Schoffers, A Golebiowski, CR Johnson Tetrahedron 52 (11), 3769-3826, 1996 | 466 | 1996 |
Development of orally bioavailable bicyclic pyrazolones as inhibitors of tumor necrosis factor-α production MP Clark, SK Laughlin, MJ Laufersweiler, RG Bookland, TA Brugel, ... Journal of medicinal chemistry 47 (11), 2724-2727, 2004 | 158 | 2004 |
Lead compounds discovered from libraries A Golebiowski, SR Klopfenstein, DE Portlock Current opinion in chemical biology 5 (3), 273-284, 2001 | 147 | 2001 |
Discovery of (R)-2-Amino-6-borono-2-(2-(piperidin-1-yl)ethyl)hexanoic Acid and Congeners As Highly Potent Inhibitors of Human Arginases I and II for Treatment of … MC Van Zandt, DL Whitehouse, A Golebiowski, MK Ji, M Zhang, ... Journal of medicinal chemistry 56 (6), 2568-2580, 2013 | 97 | 2013 |
Lead compounds discovered from libraries: part 2 A Golebiowski, SR Klopfenstein, DE Portlock Current opinion in chemical biology 7 (3), 308-325, 2003 | 96 | 2003 |
Universal Rink–isonitrile resin: application for the traceless synthesis of 3-acylamino imidazo [1, 2-a] pyridines JJ Chen, A Golebiowski, J McClenaghan, SR Klopfenstein, L West Tetrahedron Letters 42 (12), 2269-2271, 2001 | 87 | 2001 |
Synthesis of (+)-1-deoxygalactonojirimycin and a related indolizidine CR Johnson, A Golebiowski, H Sundram, MW Miller, RL Dwaihy Tetrahedron letters 36 (5), 653-654, 1995 | 87 | 1995 |
Solid supported high-throughput organic synthesis of peptide β-turn mimetics via tandem Petasis reaction/diketopiperazine formation A Golebiowski, SR Klopfenstein, JJ Chen, X Shao Tetrahedron Letters 41 (25), 4841-4844, 2000 | 84 | 2000 |
Development of new pyrrolopyrimidine-based inhibitors of Janus kinase 3 (JAK3) MP Clark, KM George, RG Bookland, J Chen, SK Laughlin, KD Thakur, ... Bioorganic & medicinal chemistry letters 17 (5), 1250-1253, 2007 | 82 | 2007 |
The development of 2-benzimidazole substituted pyrimidine based inhibitors of lymphocyte specific kinase (Lck) M Sabat, JC VanRens, MJ Laufersweiler, TA Brugel, J Maier, ... Bioorganic & medicinal chemistry letters 16 (23), 5973-5977, 2006 | 82 | 2006 |
Solid-supported synthesis of a peptide β-turn mimetic A Golebiowski, SR Klopfenstein, X Shao, JJ Chen, AO Colson, AL Grieb, ... Organic letters 2 (17), 2615-2617, 2000 | 81 | 2000 |
Synthesis of aza-C-disaccharides-a new class of sugar mimics CR Johnson, MW Miller, A Golebiowski, H Sundram, MB Ksebati Tetrahedron letters 35 (48), 8991-8994, 1994 | 78 | 1994 |
Enzymic asymmetrization in organic media: synthesis of unnatural glucose from cycloheptatriene. CR Johnson, A Golebiowski, DH Steensma Journal of the American Chemical Society 114 (24), 9414-9418, 1992 | 78 | 1992 |
Solid-supported synthesis of putative peptide β-turn mimetics via Ugi reaction for diketopiperazine formation A Golebiowski, J Jozwik, SR Klopfenstein, AO Colson, AL Grieb, ... Journal of Combinatorial Chemistry 4 (6), 584-590, 2002 | 77 | 2002 |
Automated High-Throughput Liquid− Liquid Extraction for Initial Purification of Combinatorial Libraries SX Peng, C Henson, MJ Strojnowski, A Golebiowski, SR Klopfenstein Analytical chemistry 72 (2), 261-266, 2000 | 72 | 2000 |
The development of new isoxazolone based inhibitors of tumor necrosis factor-alpha (TNF-α) production SK Laughlin, MP Clark, JF Djung, A Golebiowski, TA Brugel, M Sabat, ... Bioorganic & medicinal chemistry letters 15 (9), 2399-2403, 2005 | 67 | 2005 |
α-Amino-β-hydroxy Acids in the Total Synthesis of Amino Sugars A Gołębiowski, J Jurczak Synlett 1993 (04), 241-245, 1993 | 66 | 1993 |
Enantioselective synthesis of 6-cycloheptene-1, 3, 5-triol derivatives by enzymatic asymmetrization CR Johnson, A Golebiowski, TK McGill, DH Steensma Tetrahedron letters 32 (23), 2597-2600, 1991 | 62 | 1991 |
A practical synthesis of peptide mimetics via the solid-phase Petasis reaction SR Klopfenstein, JJ Chen, A Golebiowski, M Li, SX Peng, X Shao Tetrahedron Letters 41 (25), 4835-4839, 2000 | 60 | 2000 |