1, 4-Dihydropyridines as alkyl radical precursors: introducing the aldehyde feedstock to nickel/photoredox dual catalysis A Gutiérrez-Bonet, JC Tellis, JK Matsui, BA Vara, GA Molander ACS catalysis 6 (12), 8004-8008, 2016 | 246 | 2016 |
Scalable thioarylation of unprotected peptides and biomolecules under Ni/photoredox catalysis BA Vara, X Li, S Berritt, CR Walters, EJ Petersson, GA Molander Chemical Science 9 (2), 336-344, 2018 | 157 | 2018 |
Enantioselective small molecule synthesis by carbon dioxide fixation using a dual Brønsted acid/base organocatalyst BA Vara, TJ Struble, W Wang, MC Dobish, JN Johnston Journal of the American Chemical Society 137 (23), 7302-7305, 2015 | 127 | 2015 |
O-Benzyl Xanthate Esters under Ni/Photoredox Dual Catalysis: Selective Radical Generation and Csp3–Csp2 Cross-Coupling BA Vara, NR Patel, GA Molander ACS catalysis 7 (6), 3955-3959, 2017 | 89 | 2017 |
C (sp 3)–C (sp 2) cross-coupling of alkylsilicates with borylated aryl bromides–an iterative platform to alkylated aryl-and heteroaryl boronates BA Vara, M Jouffroy, GA Molander Chemical Science 8 (1), 530-535, 2017 | 49 | 2017 |
Organocatalytic, diastereo-and enantioselective synthesis of nonsymmetric cis-stilbene diamines: a platform for the preparation of single-enantiomer cis-imidazolines for … BA Vara, A Mayasundari, JC Tellis, MW Danneman, V Arredondo, ... The Journal of Organic Chemistry 79 (15), 6913-6938, 2014 | 49 | 2014 |
Enantioselective synthesis of β-fluoro amines via β-amino α-fluoro nitroalkanes and a traceless activating group strategy BA Vara, JN Johnston Journal of the American Chemical Society 138 (42), 13794-13797, 2016 | 45 | 2016 |
Discovery of diaminopyrimidine carboxamide HPK1 inhibitors as preclinical immunotherapy tool compounds BA Vara, SM Levi, A Achab, DA Candito, X Fradera, CA Lesburg, ... ACS Medicinal Chemistry Letters 12 (4), 653-661, 2021 | 36 | 2021 |
Reductive sp3–sp2 Coupling Reactions Enable Late-Stage Modification of Pharmaceuticals KM Mennie, BA Vara, SM Levi Organic letters 22 (2), 556-559, 2020 | 19 | 2020 |
Adaptation of a small-molecule hydrogen-bond donor catalyst to an enantioselective hetero-Diels–Alder reaction hypothesized for brevianamide biosynthesis DJ Sprague, BM Nugent, RA Yoder, BA Vara, JN Johnston Organic letters 17 (4), 880-883, 2015 | 16 | 2015 |
MDM2 antagonists counteract drug-induced DNA damage AE Vilgelm, P Cobb, K Malikayil, D Flaherty, CA Johnson, D Raman, ... EBioMedicine 24, 43-55, 2017 | 13 | 2017 |
Catal. 2016, 6, 8004–8008; d) K. Nakajima, S. Nojima, Y. Nishibayashi JC GutiØrrez-Bonet, JK Tellis, BA Matsui, GA Vara, ACS Molander Angew. Chem. Int. Ed 55, 14106-14110, 2016 | 12 | 2016 |
The n-dig-Cyclization (n= 5, 6) of Alkynes Involving Fixation of CO2 B Wang, S Sun, J Cheng Synlett 29 (14), 1814-1822, 2018 | 6 | 2018 |
Activation of hepatocyte growth factor/MET signaling as a mechanism of acquired resistance to a novel YAP1/TEAD small molecule inhibitor CJ Moure, B Vara, MM Cheng, C Sondey, E Muise, E Park, ... Molecular Cancer Therapeutics 23 (8), 1095-1108, 2024 | 1 | 2024 |
Diaminopyrimidine carboxamide inhibitors of hpk1 A Achab, DA Candito, A Donofrio, X Fradera, S Kawamura, SM Levi, B Li, ... US Patent App. 18/251,259, 2023 | 1 | 2023 |
Assessment of a receptor-interacting serine/threonine-protein kinase 1 (RIPK1) PET tracer feasibility:[18F] A in in vitro brain tissue based binding assay and in vivo PET … W Li, B Vara, D Rubins, P Dockery, K Riffel, Y Wang, Z Zeng, C Sondey, ... Journal of Nuclear Medicine 65 (supplement 2), 242075-242075, 2024 | | 2024 |
Aryl ether compounds as tead modulators J Lim, V Simov, BA Vara, CS Yeung, SE Schneider, EF DiMauro US Patent App. 18/264,468, 2024 | | 2024 |
Ripk1 inhibitors and methods of use JL Chen, YH Chen, EF DiMauro, M Liu, JL Methot, AJ Musacchio, ... US Patent App. 18/318,760, 2024 | | 2024 |
7-phenyl substituted 2-aminoquinazoline inhibitors of hpk1 DA Candito, JL Chen, A Donofrio, X Fradera, PH Fuller, S Kawamura, B Li, ... US Patent App. 18/250,419, 2023 | | 2023 |
Spirotricycle ripk1 inhibitors and methods of uses thereof AA Achab, ZG Brill, JLR Duque, X Fradera, JL Methot, P Siliphaivanh, ... US Patent App. 18/049,344, 2023 | | 2023 |