Stefan Knapp

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388 articoli

66 articoli

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Panagis FilippakopoulosAssociate Professor, Oxford UniversityEmail verificata su sgc.ox.ac.uk
Oleg FedorovUniversity of OxfordEmail verificata su cmd.ox.ac.uk
Apirat ChaikuadEmail verificata su pharmchem.uni-frankfurt.de
Paul E BrennanUniversity of OxfordEmail verificata su cmd.ox.ac.uk
Frank von DelftPrincipal Investigator: Protein Crystallography, SGC, Oxford UniversityEmail verificata su sgc.ox.ac.uk
Brian MarsdenCentre for Medicines Discovery & Centre for Human Genetics, NDM, University of OxfordEmail verificata su cmd.ox.ac.uk
Sebastian MatheaEmail verificata su pharmchem.uni-frankfurt.de
Wen Hwa LeeAction Against AMD, SGC and University of OxfordEmail verificata su actionagainstamd.org
Cheryl ArrowsmithSenior Scientist, Princess Margaret Cancer Centre & Professor of Medical Biophysics, University of TorontoEmail verificata su uhnres.utoronto.ca
Benjamin E. TurkYale UniversityEmail verificata su yale.edu
Jeyanthy EswaranSaint Jude's Children's Research HospitalEmail verificata su stjude.org
Chas BountraProfessor of Translational MedicineEmail verificata su cmd.ox.ac.uk
Martin SchröderNovartis Institute for Biomedical ResearchEmail verificata su novartis.com
Opher GileadiSGC, Karolinska InstituteEmail verificata su ki.se
Juerg SchwallerProfessor Universität BaselEmail verificata su unibas.ch
Ashley PikeCentre for Medicines Discovery - University of OxfordEmail verificata su cmd.ox.ac.uk
Kilian V. M. HuberPrincipal Investigator, University of OxfordEmail verificata su cmd.ox.ac.uk
Stuart J ConwayJung Chair in Medicinal Chemistry, University of California, Los AngelesEmail verificata su chem.ucla.edu
Laurent MeijerEmail verificata su manros-therapeutics.com
David Harold DrewryProfessor University of North Carolina Chapel HillEmail verificata su unc.edu

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Stefan Knapp

University of Frankfurt

Email verificata su pharmchem.uni-frankfurt.de

bromodomains kinases structural biology drug design


Titolo Ordina per citazioni Ordina per anno Ordina per titolo	Citata da Citata da	Anno
Selective inhibition of BET bromodomains P Filippakopoulos, J Qi, S Picaud, Y Shen, WB Smith, O Fedorov, ... Nature 468 (7327), 1067-1073, 2010	4433	2010
Histone recognition and large-scale structural analysis of the human bromodomain family P Filippakopoulos, S Picaud, M Mangos, T Keates, JP Lambert, ... Cell 149 (1), 214-231, 2012	1800	2012
Targeting bromodomains: epigenetic readers of lysine acetylation P Filippakopoulos, S Knapp Nature reviews Drug discovery 13 (5), 337-356, 2014	1351	2014
Protein production and purification Architecture et Fonction des Macromolécules Biologiques Vincentelli Renaud 4 ... Nature methods 5 (2), 135-146, 2008	1030	2008
The promise and peril of chemical probes CH Arrowsmith, JE Audia, C Austin, J Baell, J Bennett, J Blagg, C Bountra, ... Nature chemical biology 11 (8), 536-541, 2015	863	2015
Critical residues for structure and catalysis in short-chain dehydrogenases/reductases C Filling, KD Berndt, J Benach, S Knapp, T Prozorovski, E Nordling, ... Journal of Biological Chemistry 277 (28), 25677-25684, 2002	687	2002
The molecular mechanism of nitrogen-containing bisphosphonates as antiosteoporosis drugs KL Kavanagh, K Guo, JE Dunford, X Wu, S Knapp, FH Ebetino, ... Proceedings of the National Academy of Sciences 103 (20), 7829-7834, 2006	669	2006
Bromodomains as therapeutic targets S Muller, P Filippakopoulos, S Knapp Expert reviews in molecular medicine 13, e29, 2011	559	2011
Copper is required for oncogenic BRAF signalling and tumorigenesis DC Brady, MS Crowe, ML Turski, GA Hobbs, X Yao, A Chaikuad, S Knapp, ... Nature 509 (7501), 492-496, 2014	555	2014
Large-scale structural analysis of the classical human protein tyrosine phosphatome AJ Barr, E Ugochukwu, WH Lee, ONF King, P Filippakopoulos, I Alfano, ... Cell 136 (2), 352-363, 2009	553	2009
Trends in kinase drug discovery: targets, indications and inhibitor design MM Attwood, D Fabbro, AV Sokolov, S Knapp, HB Schiöth Nature Reviews Drug Discovery 20 (11), 839-861, 2021	534	2021
Linear motif atlas for phosphorylation-dependent signaling ML Miller, LJ Jensen, F Diella, C Jørgensen, M Tinti, L Li, M Hsiung, ... Science signaling 1 (35), ra2-ra2, 2008	534	2008
Small-molecule inhibition of BRDT for male contraception MM Matzuk, MR McKeown, P Filippakopoulos, Q Li, L Ma, JE Agno, ... Cell 150 (4), 673-684, 2012	522	2012
RVX-208, an inhibitor of BET transcriptional regulators with selectivity for the second bromodomain S Picaud, C Wells, I Felletar, D Brotherton, S Martin, P Savitsky, ... Proceedings of the National Academy of Sciences 110 (49), 19754-19759, 2013	496	2013
The bromodomain interaction module P Filippakopoulos, S Knapp FEBS letters 586 (17), 2692-2704, 2012	464	2012
Stereospecific targeting of MTH1 by (S)-crizotinib as an anticancer strategy KVM Huber, E Salah, B Radic, M Gridling, JM Elkins, A Stukalov, ... Nature 508 (7495), 222-227, 2014	452	2014
Exploration of type II binding mode: A privileged approach for kinase inhibitor focused drug discovery? Z Zhao, H Wu, L Wang, Y Liu, S Knapp, Q Liu, NS Gray ACS chemical biology 9 (6), 1230-1241, 2014	434	2014
PIM serine/threonine kinases in the pathogenesis and therapy of hematologic malignancies and solid cancers L Brault, C Gasser, F Bracher, K Huber, S Knapp, J Schwaller haematologica 95 (6), 1004, 2010	431	2010
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases O Fedorov, B Marsden, V Pogacic, P Rellos, S Müller, AN Bullock, ... Proceedings of the National Academy of Sciences 104 (51), 20523-20528, 2007	420	2007
Crystal structure of the tetrameric Mad1–Mad2 core complex: implications of a ‘safety belt’binding mechanism for the spindle checkpoint L Sironi, M Mapelli, S Knapp, A De Antoni, KT Jeang, A Musacchio The EMBO journal, 2002	396	2002

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