Articoli con mandati relativi all'accesso pubblico - James BradnerUlteriori informazioni
Non disponibili pubblicamente: 3
PRC2 loss amplifies Ras-driven transcription and confers sensitivity to BRD4-based therapies
T De Raedt, E Beert, E Pasmant, A Luscan, H Brems, N Ortonne, K Helin, ...
Nature 514 (7521), 247-251, 2014
Mandati: US National Institutes of Health, Research Foundation (Flanders), National …
Translation termination factor GSPT1 is a phenotypically relevant off-target of heterobifunctional phthalimide degraders
M Ishoey, S Chorn, N Singh, MG Jaeger, M Brand, J Paulk, S Bauer, ...
ACS Chemical Biology 13 (3), 553-560, 2018
Mandati: US National Institutes of Health, Carlsberg Foundation DK
A chemical probe toolbox for dissecting the cancer epigenome
J Shortt, CJ Ott, RW Johnstone, JE Bradner
Nature Reviews Cancer 17 (3), 160-183, 2017
Mandati: US National Institutes of Health, National Health and Medical Research …
Disponibili pubblicamente: 247
Selective inhibition of BET bromodomains
P Filippakopoulos, J Qi, S Picaud, Y Shen, WB Smith, O Fedorov, ...
Nature 468 (7327), 1067-1073, 2010
Mandati: US National Institutes of Health, Canadian Institutes of Health Research …
BET bromodomain inhibition as a therapeutic strategy to target c-Myc
JE Delmore, GC Issa, ME Lemieux, PB Rahl, J Shi, HM Jacobs, E Kastritis, ...
Cell 146 (6), 904-917, 2011
Mandati: US National Institutes of Health
Selective inhibition of tumor oncogenes by disruption of super-enhancers
J Lovén, HA Hoke, CY Lin, A Lau, DA Orlando, CR Vakoc, JE Bradner, ...
Cell 153 (2), 320-334, 2013
Mandati: US National Institutes of Health, Swedish Research Council
RNAi screen identifies Brd4 as a therapeutic target in acute myeloid leukaemia
J Zuber, J Shi, E Wang, AR Rappaport, H Herrmann, EA Sison, D Magoon, ...
Nature 478 (7370), 524-528, 2011
Mandati: US National Institutes of Health, Howard Hughes Medical Institute, German …
HDAC2 negatively regulates memory formation and synaptic plasticity
JS Guan, SJ Haggarty, E Giacometti, JH Dannenberg, N Joseph, J Gao, ...
Nature 459 (7243), 55-60, 2009
Mandati: US National Institutes of Health, Howard Hughes Medical Institute
Transcriptional amplification in tumor cells with elevated c-Myc
CY Lin, J Lovén, PB Rahl, RM Paranal, CB Burge, JE Bradner, TI Lee, ...
Cell 151 (1), 56-67, 2012
Mandati: US National Institutes of Health, Swedish Research Council
Phthalimide conjugation as a strategy for in vivo target protein degradation
GE Winter, DL Buckley, J Paulk, JM Roberts, A Souza, S Dhe-Paganon, ...
Science 348 (6241), 1376-1381, 2015
Mandati: US National Institutes of Health, John D. and Catherine T. MacArthur …
The myeloma drug lenalidomide promotes the cereblon-dependent destruction of Ikaros proteins
G Lu, RE Middleton, H Sun, MV Naniong, CJ Ott, CS Mitsiades, KK Wong, ...
Science 343 (6168), 305-309, 2014
Mandati: US National Institutes of Health, Howard Hughes Medical Institute, German …
Transcriptional addiction in cancer
JE Bradner, D Hnisz, RA Young
Cell 168 (4), 629-643, 2017
Mandati: US National Institutes of Health, Austrian Science Fund
R-2HG exhibits anti-tumor activity by targeting FTO/m6A/MYC/CEBPA signaling
R Su, L Dong, C Li, S Nachtergaele, M Wunderlich, Y Qing, X Deng, ...
Cell 172 (1), 90-105. e23, 2018
Mandati: US National Institutes of Health, Howard Hughes Medical Institute, Damon …
Direct inhibition of the NOTCH transcription factor complex
RE Moellering, M Cornejo, TN Davis, CD Bianco, JC Aster, SC Blacklow, ...
Nature 462 (7270), 182-188, 2009
Mandati: US National Institutes of Health
YY1 is a structural regulator of enhancer-promoter loops
AS Weintraub, CH Li, AV Zamudio, AA Sigova, NM Hannett, DS Day, ...
Cell 171 (7), 1573-1588. e28, 2017
Mandati: US National Science Foundation, US National Institutes of Health, Damon …
Chemical phylogenetics of histone deacetylases
JE Bradner, N West, ML Grachan, EF Greenberg, SJ Haggarty, T Warnow, ...
Nature chemical biology 6 (3), 238-243, 2010
Mandati: US National Institutes of Health
Discovery and characterization of super-enhancer-associated dependencies in diffuse large B cell lymphoma
B Chapuy, MR McKeown, CY Lin, S Monti, MGM Roemer, J Qi, PB Rahl, ...
Cancer cell 24 (6), 777-790, 2013
Mandati: US National Institutes of Health, German Research Foundation
The dTAG system for immediate and target-specific protein degradation
B Nabet, JM Roberts, DL Buckley, J Paulk, S Dastjerdi, A Yang, ...
Nature chemical biology 14 (5), 431-441, 2018
Mandati: US National Institutes of Health, Damon Runyon Cancer Research Foundation
A single oncogenic enhancer rearrangement causes concomitant EVI1 and GATA2 deregulation in leukemia
S Gröschel, MA Sanders, R Hoogenboezem, E de Wit, BAM Bouwman, ...
Cell 157 (2), 369-381, 2014
Mandati: German Research Foundation, Worldwide Cancer Research, UK
Targeting MYCN in neuroblastoma by BET bromodomain inhibition
A Puissant, SM Frumm, G Alexe, CF Bassil, J Qi, YH Chanthery, ...
Cancer discovery 3 (3), 308-323, 2013
Mandati: US National Institutes of Health, Howard Hughes Medical Institute
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