| Azaindoles: Noncovalent DprE1 Inhibitors from Scaffold Morphing Efforts, Kill Mycobacterium tuberculosis and Are Efficacious in Vivo PS Shirude, R Shandil, C Sadler, M Naik, V Hosagrahara, S Hameed, ... Journal of Medicinal Chemistry 56 (23), 9701-9708, 2013 | 173 | 2013 |
| Discovery of Imidazo[1,2-a]pyridine Ethers and Squaramides as Selective and Potent Inhibitors of Mycobacterial Adenosine Triphosphate (ATP) Synthesis SJ Tantry, SD Markad, V Shinde, J Bhat, G Balakrishnan, AK Gupta, ... Journal of medicinal chemistry 60 (4), 1379-1399, 2017 | 130 | 2017 |
| 1, 4-Azaindole, a potential drug candidate for treatment of tuberculosis M Chatterji, R Shandil, MR Manjunatha, S Solapure, V Ramachandran, ... Antimicrobial agents and chemotherapy 58 (9), 5325-5331, 2014 | 118 | 2014 |
| Lead optimization of 1, 4-azaindoles as antimycobacterial agents PS Shirude, RK Shandil, MR Manjunatha, C Sadler, M Panda, V Panduga, ... Journal of medicinal chemistry 57 (13), 5728-5737, 2014 | 113 | 2014 |
| 4-aminoquinolone piperidine amides: noncovalent inhibitors of DprE1 with long residence time and potent antimycobacterial activity M Naik, V Humnabadkar, SJ Tantry, M Panda, A Narayan, S Guptha, ... Journal of medicinal chemistry 57 (12), 5419-5434, 2014 | 105 | 2014 |
| In Vitro and In Vivo Efficacy of β-Lactams against Replicating and Slowly Growing/Nonreplicating Mycobacterium tuberculosis S Solapure, N Dinesh, R Shandil, V Ramachandran, S Sharma, ... Antimicrobial agents and chemotherapy 57 (6), 2506-2510, 2013 | 85 | 2013 |
| Triaminopyrimidine is a fast-killing and long-acting antimalarial clinical candidate S Hameed P, S Solapure, V Patil, PP Henrich, PA Magistrado, S Bharath, ... Nature Communications 6 (1), 6715, 2015 | 81 | 2015 |
| Thiazolopyridine ureas as novel antitubercular agents acting through inhibition of DNA gyrase B MG Kale, A Raichurkar, SH P, D Waterson, D McKinney, MR Manjunatha, ... Journal of medicinal chemistry 56 (21), 8834-8848, 2013 | 71 | 2013 |
| Benzimidazoles: novel mycobacterial gyrase inhibitors from scaffold morphing S Hameed P, A Raichurkar, P Madhavapeddi, S Menasinakai, S Sharma, ... ACS Medicinal Chemistry Letters 5 (7), 820-825, 2014 | 59 | 2014 |
| Novel N-Linked Aminopiperidine-Based Gyrase Inhibitors with Improved hERG and in Vivo Efficacy against Mycobacterium tuberculosis S Hameed P, V Patil, S Solapure, U Sharma, P Madhavapeddi, ... Journal of Medicinal Chemistry 57 (11), 4889-4905, 2014 | 50 | 2014 |
| Whole cell screen based identification of spiropiperidines with potent antitubercular properties SJ Tantry, G Degiacomi, S Sharma, L kumar Jena, A Narayan, S Guptha, ... Bioorganic & medicinal chemistry letters 25 (16), 3234-3245, 2015 | 47 | 2015 |
| Optimization of pyrrolamides as mycobacterial GyrB ATPase inhibitors: structure-activity relationship and in vivo efficacy in a mouse model of tuberculosis S Solapure, K Mukherjee, V Nandi, D Waterson, R Shandil, M Balganesh, ... Antimicrobial agents and chemotherapy 58 (1), 61, 2014 | 46 | 2014 |
| N-Aryl-2-aminobenzimidazoles: Novel, Efficacious, Antimalarial Lead Compounds S Ramachandran, S Hameed P, A Srivastava, G Shanbhag, S Morayya, ... Journal of Medicinal Chemistry 57 (15), 6642-6652, 2014 | 45 | 2014 |
| A comparison of sorghum stover based complete feed blocks with a conventional feeding practice in a peri urban dairy S Anandan, AA Khan, D Ravi, J Reddy, M Blümmel Animal Nutrition and Feed Technology 10 (spl), 23-28, 2010 | 38 | 2010 |
| Aminoazabenzimidazoles, a novel class of orally active antimalarial agents S Hameed P, M Chinnapattu, G Shanbag, P Manjrekar, K Koushik, ... Journal of Medicinal Chemistry 57 (13), 5702-5713, 2014 | 34 | 2014 |
| Effect of coadministration of moxifloxacin and rifampin on Mycobacterium tuberculosis in a murine aerosol infection model V Balasubramanian, S Solapure, S Gaonkar, KN Mahesh Kumar, ... Antimicrobial agents and chemotherapy 56 (6), 3054-3057, 2012 | 34 | 2012 |
| Pharmacokinetics and dose response of anti-TB drugs in rat infection model of tuberculosis N Kumar, KG Vishwas, M Kumar, J Reddy, M Parab, CL Manikanth, ... Tuberculosis 94 (3), 282-286, 2014 | 31 | 2014 |
| Scaffold morphing leading to evolution of 2, 4-diaminoquinolines and aminopyrazolopyrimidines as inhibitors of the ATP synthesis pathway SJ Tantry, V Shinde, G Balakrishnan, SD Markad, AK Gupta, J Bhat, ... MedChemComm 7 (5), 1022-1032, 2016 | 30 | 2016 |
| Pharmacokinetic and pharmacodynamic evaluation of AZD5847 in a mouse model of tuberculosis V Balasubramanian, S Solapure, R Shandil, S Gaonkar, KN Mahesh, ... Antimicrobial agents and chemotherapy 58 (7), 4185-4190, 2014 | 25 | 2014 |
| Ammonium iodide-mediated sulfenylation of 4-hydroxycoumarins or 4-hydroxyquinolinones with a sulfonyl chloride as a sulfur source T Guo, XN Wei Synlett 28 (18), 2499-2504, 2017 | 24 | 2017 |