Metathesis in the synthesis of aromatic compounds WAL van Otterlo, CB De Koning Chemical reviews 109 (8), 3743-3782, 2009 | 317 | 2009 |
Isomerization of allylbenzenes M Hassam, A Taher, GE Arnott, IR Green, WAL van Otterlo Chemical reviews 115 (11), 5462-5569, 2015 | 289 | 2015 |
Modern methods for the synthesis of substituted naphthalenes CB de Koning, AL Rousseau, WAL van Otterlo Tetrahedron 59 (1), 7-36, 2003 | 235 | 2003 |
Bioactivity-guided mapping and navigation of chemical space S Renner, WAL Van Otterlo, M Dominguez Seoane, S Möcklinghoff, ... Nature chemical biology 5 (8), 585-592, 2009 | 162 | 2009 |
Ring-closing metathesis for the synthesis of 2H-and 4H-chromenes WAL Van Otterlo, EL Ngidi, S Kuzvidza, GL Morgans, SS Moleele, ... Tetrahedron 61 (42), 9996-10006, 2005 | 132 | 2005 |
The synthesis of 2-and 3-aryl indoles and 1, 3, 4, 5-tetrahydropyrano [4, 3-b] indoles and their antibacterial and antifungal activity TC Leboho, JP Michael, WAL van Otterlo, SF van Vuuren, CB de Koning Bioorganic & medicinal chemistry letters 19 (17), 4948-4951, 2009 | 120 | 2009 |
An isomerization-ring-closing metathesis strategy for the synthesis of substituted benzofurans WAL van Otterlo, GL Morgans, LG Madeley, S Kuzvidza, SS Moleele, ... Tetrahedron 61 (32), 7746-7755, 2005 | 120 | 2005 |
Covalent‐allosteric kinase inhibitors J Weisner, R Gontla, L van der Westhuizen, S Oeck, J Ketzer, P Janning, ... Angewandte Chemie International Edition 54 (35), 10313-10316, 2015 | 111 | 2015 |
Sequential isomerization and ring-closing metathesis: masked styryl and vinyloxyaryl groups for the synthesis of benzo-fused heterocycles WAL van Otterlo, EL Ngidi, CB de Koning Tetrahedron letters 44 (34), 6483-6486, 2003 | 98 | 2003 |
Synthesis and biological evaluation of 4-anilinoquinolines as potent inhibitors of epidermal growth factor receptor VG Pawar, ML Sos, HB Rode, M Rabiller, S Heynck, WAL Van Otterlo, ... Journal of medicinal chemistry 53 (7), 2892-2901, 2010 | 93 | 2010 |
In search of a treatment for HIV–current therapies and the role of non-nucleoside reverse transcriptase inhibitors (NNRTIs) C Reynolds, CB de Koning, SC Pelly, WAL van Otterlo, ML Bode Chemical Society Reviews 41 (13), 4657-4670, 2012 | 92 | 2012 |
Toward a cancer drug of fungal origin A Kornienko, A Evidente, M Vurro, V Mathieu, A Cimmino, M Evidente, ... Medicinal research reviews 35 (5), 937-967, 2015 | 89 | 2015 |
Isomerization and ring-closing metathesis for the synthesis of 6-, 7-and 8-membered benzo-and pyrido-fused N, N-, N, O-and N, S-heterocycles WAL van Otterlo, GL Morgans, SD Khanye, BAA Aderibigbe, JP Michael, ... Tetrahedron letters 45 (50), 9171-9175, 2004 | 88 | 2004 |
Metathesis reactions for the synthesis of ring-fused carbazoles SC Pelly, CJ Parkinson, WAL Van Otterlo, CB De Koning The Journal of Organic Chemistry 70 (25), 10474-10481, 2005 | 87 | 2005 |
Synthesis of the dibenzopyrrocoline alkaloid skeleton: indolo [2, 1-a] isoquinolines and related analogues ANC Lötter, R Pathak, TS Sello, MA Fernandes, WAL van Otterlo, ... Tetrahedron 63 (10), 2263-2274, 2007 | 84 | 2007 |
Ring-closing metathesis for the synthesis of benzo-fused bicyclic compounds WAL van Otterlo, EL Ngidi, EM Coyanis, CB de Koning Tetrahedron letters 44 (2), 311-313, 2003 | 83 | 2003 |
Conjugated polymer stabilized palladium nanoparticles as a versatile catalyst for Suzuki cross-coupling reactions for both aryl and heteroaryl bromide systems RU Islam, MJ Witcomb, MS Scurrell, E Van Der Lingen, W Van Otterlo, ... Catalysis Science & Technology 1 (2), 308-315, 2011 | 76 | 2011 |
A concise synthesis of novel naphtho [a] carbazoles and benzo [c] carbazoles R Pathak, JM Nhlapo, S Govender, JP Michael, WAL van Otterlo, ... Tetrahedron 62 (12), 2820-2830, 2006 | 75 | 2006 |
In search of a cytostatic agent derived from the alkaloid lycorine: Synthesis and growth inhibitory properties of lycorine derivatives NM Evdokimov, D Lamoral-Theys, V Mathieu, A Andolfi, LV Frolova, ... Bioorganic & medicinal chemistry 19 (23), 7252-7261, 2011 | 69 | 2011 |
Anticancer properties of an important drug lead podophyllotoxin can be efficiently mimicked by diverse heterocyclic scaffolds accessible via one-step synthesis IV Magedov, L Frolova, M Manpadi, U Bhoga, H Tang, NM Evdokimov, ... Journal of medicinal chemistry 54 (12), 4234-4246, 2011 | 66 | 2011 |