An Easy Access to 4, 5‐Disubstituted Thiazoles via Base‐Induced Click Reaction of Active Methylene Isocyanides with Methyl Dithiocarboxylates. GS Lingaraju, TR Swaroop, AC Vinayaka, KSS Kumar, MP Sadashiva, ... ChemInform 43 (36), 2012 | 102 | 2012 |
Synthesis and microbial inhibition study of novel 5-imidazolyl substituted isoxazolidines MP Sadashiva, H Mallesha, NA Hitesh, KS Rangappa Bioorganic & medicinal chemistry 12 (24), 6389-6395, 2004 | 76 | 2004 |
A hirshfeld surface analysis and crystal structure of 2'-1-(2-fluoro-phenyl)-1H-tetrazol-5-Yl-4-methoxy-biphenyl-2-carbaldehyde S Madan Kumar, BC Manjunath, GS Lingaraju, MMM Abdoh, ... Crystal Structure Theory and Applications 2 (3), 124-131, 2013 | 63 | 2013 |
Synthesis of new coumarin tethered isoxazolines as potential anticancer agents GS Lingaraju, KS Balaji, S Jayarama, SM Anil, KR Kiran, MP Sadashiva Bioorganic & medicinal chemistry letters 28 (23-24), 3606-3612, 2018 | 62 | 2018 |
Anti-cancer activity of novel dibenzo [b, f] azepine tethered isoxazoline derivatives MP Sadashiva, Basappa, S NanjundaSwamy, F Li, KA Manu, ... BMC Chemical Biology 12, 5, 2012 | 57 | 2012 |
Solution-phase synthesis of novel Δ2-isoxazoline libraries via 1, 3-dipolar cycloaddition and their antifungal properties MP Sadashiva, K Mantelingu, SN Swamy, KS Rangappa Bioorganic & medicinal chemistry 11 (21), 4539-4544, 2003 | 57 | 2003 |
Facile synthesis of 1, 4-benzodiazepine-2, 5-diones and quinazolinones from amino acids as anti-tubercular agents SM Anil, R Shobith, KR Kiran, TR Swaroop, N Mallesha, MP Sadashiva New Journal of Chemistry 43 (1), 182-187, 2019 | 51 | 2019 |
Weinreb amide as an efficient reagent in the one pot synthesis of benzimidazoles and benzothiazoles YK Bommegowda, GS Lingaraju, S Thamas, KSV Kumar, CSP Kumara, ... Tetrahedron Letters 54 (21), 2693-2695, 2013 | 47 | 2013 |
Enhancement in antimicrobial activity of 2-(phenyl)-3-(2-butyl-4-chloro-1H-imidazolyl)-5-butylate isoxazolidine MP Sadashiva, H Mallesha, KK Murthy, KS Rangappa Bioorganic & medicinal chemistry letters 15 (7), 1811-1814, 2005 | 45 | 2005 |
A new ibuprofen derivative inhibits platelet aggregation and ROS mediated platelet apoptosis KS Rakesh, S Jagadish, AC Vinayaka, M Hemshekhar, M Paul, ... PloS one 9 (9), e107182, 2014 | 44 | 2014 |
Cyclization of active methylene isocyanides with α-oxodithioesters induced by base: An expedient synthesis of 4-methylthio/ethoxycarbonyl-5-acylthiazoles KR Kiran, TR Swaroop, N Rajeev, SM Anil, KS Rangappa, MP Sadashiva Synthesis 52 (09), 1444-1450, 2020 | 41 | 2020 |
Platelet protective efficacy of 3, 4, 5 trisubstituted isoxazole analogue by inhibiting ROS-mediated apoptosis and platelet aggregation S Jagadish, N Rajeev, SK NaveenKumar, KS Sharath Kumar, M Paul, ... Molecular and cellular biochemistry 414, 137-151, 2016 | 31 | 2016 |
Acid-Catalyzed Condensation of o-Phenylenediammines and o-Aminophenols with α-Oxodithioesters: A Divergent and Regioselective Synthesis of 2-Methylthio-3-aryl … KR Kiran, TR Swaroop, KP Sukrutha, JB Shruthi, SM Anil, KS Rangappa, ... Synthesis 51 (22), 4205-4214, 2019 | 30 | 2019 |
A simple and efficient method for the synthesis of 1, 2-benzisoxazoles: a series of its potent acetylcholinesterase inhibitors K Mantelingu, MP Sadashiva, KS Rangappa NISCAIR-CSIR, India, 2004 | 30 | 2004 |
Base-Induced Cyclization of active methylene isocyanides with xanthate esters: an efficient method for the synthesis of 5-Alkoxy-4-(tosyl/ethoxycarbonyl)-1, 3-thiazoles N Rajeev, TR Swaroop, SM Anil, YK Bommegowda, KS Rangappa, ... Synlett 28 (17), 2281-2284, 2017 | 28 | 2017 |
Transition-metal-free solid phase synthesis of 1,2-disubstituted 4-quinolones via regiospecific synthesis of enaminones KSRMPS Ajjampura C Vinayaka, Toreshettahally R Swaroop, Prasanna Kumara Chikkade RSC Adv.,, 2016 | 28 | 2016 |
Green Photoorganocatalytic Synthesis of Phenols from Arylboronic Acids IK Sideri, E Voutyritsa, CG Kokotos Synlett 29 (10), 1324-1328, 2018 | 27 | 2018 |
Facile synthesis of antimalarial 1, 2-disubstituted 4-quinolones from 1, 3-bisaryl-monothio-1, 3-diketones AC Vinayaka, MP Sadashiva, X Wu, SS Biryukov, JA Stoute, ... Organic & Biomolecular Chemistry 12 (42), 8555-8561, 2014 | 27 | 2014 |
The regioselective synthesis of 2, 5-and 4, 5-disubstituted thiazoles via the cyclization of 2-oxo-2-(amino) ethanedithioates with isocyanides KR Singh, C Santhosh, TR Swaroop, MP Sadashiva Organic & Biomolecular Chemistry 20 (29), 5771-5778, 2022 | 26 | 2022 |
A one-pot tandem approach for the synthesis of 5-(het) aryloxazoles from substituted (het) aryl methyl alcohols and benzyl bromides KSV Kumar, TR Swaroop, N Rajeev, AC Vinayaka, GS Lingaraju, ... Synlett 27 (09), 1363-1366, 2016 | 26 | 2016 |