Stereoselective Formal [3 + 3] Cycloaddition Approach to cis-1-Azadecalins and Synthesis of (−)-4a,8a-diepi-Pumiliotoxin C. Evidence for the First Highly … HM Sklenicka, RP Hsung, MJ McLaughlin, L Wei, AI Gerasyuto, ... Journal of the American Chemical Society 124 (35), 10435-10442, 2002 | 122 | 2002 |
A Novel and Highly Stereoselective Intramolecular Formal [3+3] Cycloaddition Reaction of Vinylogous Amides Tethered with α,β‐Unsaturated Aldehydes: A … LL Wei, RP Hsung, HM Sklenicka, AI Gerasyuto Angewandte Chemie 113 (8), 1564-1566, 2001 | 116 | 2001 |
A formal [3+ 3] cycloaddition reaction. 5. An enantioselective intramolecular formal aza-[3+ 3] cycloaddition reaction promoted by chiral amine salts AI Gerasyuto, RP Hsung, N Sydorenko, B Slafer The Journal of Organic Chemistry 70 (11), 4248-4256, 2005 | 86 | 2005 |
A formal [3+ 3] cycloaddition reaction. improved reactivity using α, β-unsaturated iminium salts and evidence for reversibility of 6π-electron electrocyclic ring closure of 1 … HC Shen, J Wang, KP Cole, MJ McLaughlin, CD Morgan, CJ Douglas, ... The Journal of Organic Chemistry 68 (5), 1729-1735, 2003 | 85 | 2003 |
Highly Stereoselective Formal [3+ 3] Cycloaddition Reactions of Chiral Vinylogous Amides with α, β-Unsaturated Iminiums HM Sklenicka, RP Hsung, LL Wei, MJ McLaughlin, AI Gerasyuto, ... Organic Letters 2 (8), 1161-1164, 2000 | 68 | 2000 |
An Intramolecular aza-[3 + 3] Annulation Approach to Azaphenalene Alkaloids. Total Synthesis of Myrrhine AI Gerasyuto, RP Hsung The Journal of Organic Chemistry 72 (7), 2476-2484, 2007 | 45 | 2007 |
Total syntheses of enantiomerically enriched R-(+)-and S-(−)-deplancheine N Sydorenko, CA Zificsak, AI Gerasyuto, RP Hsung Organic & Biomolecular Chemistry 3 (11), 2140-2144, 2005 | 41 | 2005 |
Stereodivergent total syntheses of precoccinelline, hippodamine, coccinelline, and convergine AI Gerasyuto, RP Hsung Organic Letters 8 (21), 4899-4902, 2006 | 39 | 2006 |
Potent antimalarials with development potential identified by structure-guided computational optimization of a pyrrole-based dihydroorotate dehydrogenase inhibitor series MJ Palmer, X Deng, S Watts, G Krilov, A Gerasyuto, S Kokkonda, ... Journal of medicinal chemistry 64 (9), 6085-6136, 2021 | 35 | 2021 |
Asymmetric Aza-[3 + 3] Annulation in the Synthesis of Indolizidines: An Unexpected Reversal of Regiochemistry GS Buchanan, H Dai, RP Hsung, AI Gerasyuto, CM Scheinebeck Organic letters 13 (16), 4402-4405, 2011 | 31 | 2011 |
Organocatalyzed [3+ 3] Annulations for the Construction of Heterocycles Y Zhu, Y Huang Synthesis 52 (08), 1181-1202, 2020 | 27 | 2020 |
Inhibitors of (alpha-v)(beta-6) integrin BA Harrison, MG Bursavich, M Brewer, AI Gerasyuto, KN Hahn, KD Konze, ... US Patent App. 15/906,745, 2018 | 19 | 2018 |
Ribonucleotide reductase, a novel drug target for gonorrhea J Narasimhan, S Letinski, SP Jung, A Gerasyuto, J Wang, M Arnold, ... Elife 11, e67447, 2022 | 14 | 2022 |
Discovery and optimization of indolyl-containing 4-hydroxy-2-pyridone type II DNA topoisomerase inhibitors active against multidrug resistant gram-negative bacteria AI Gerasyuto, MA Arnold, J Wang, G Chen, X Zhang, S Smith, MG Woll, ... Journal of medicinal chemistry 61 (10), 4456-4475, 2018 | 14 | 2018 |
Synthesis of 2, 3-Dihydrobenzothiazol-1, 1-dioxide and 2, 3-Dihydro-1, 4-benzothiazin-3-one Nitroderivatives from 2, 4-Di-and 2, 4, 6-Trinitrobenzamides AI Gerasyuto, SG Zlotin, VV Semenov Synthesis 2001 (02), 0300-0304, 2001 | 12 | 2001 |
4-Hydroxy-2-pyridones: Discovery and evaluation of a novel class of antibacterial agents targeting DNA synthesis MA Arnold, AI Gerasyuto, J Wang, W Du, YJK Gorske, T Arasu, J Baird, ... Bioorganic & Medicinal Chemistry Letters 27 (22), 5014-5021, 2017 | 9 | 2017 |
Inhibiting (alpha-v)(beta-6) integrin BA Harrison, JE Dowling, MG Bursavich, DM Troast, BS Lippa, BN Rogers, ... US Patent App. 16/555,589, 2020 | 8 | 2020 |
Establishing the concept of aza-[3+ 3] annulations using enones as a key expansion of this unified strategy in alkaloid synthesis AI Gerasyuto, ZX Ma, GS Buchanan, RP Hsung Beilstein Journal of Organic Chemistry 9 (1), 1170-1178, 2013 | 8 | 2013 |
Inhibitors of (α-v)(β-6) integrin BA Harrison, MG Bursavich, M Brewer, AI Gerasyuto, KN Hahn, KD Konze, ... US Patent 11,046,669, 2021 | 7 | 2021 |
Inhibitors of (α-v)(β-6) integrin BA Harrison, MG Bursavich, AI Gerasyuto, KN Hahn, KD Konze, FY Lin, ... US Patent 11,046,685, 2021 | 7 | 2021 |