Targeting matrix metalloproteinases: Exploring the dynamics of the S1′ pocket in the design of selective, small molecule inhibitors: Miniperspective B Fabre, A Ramos, B de Pascual-Teresa Journal of medicinal chemistry 57 (24), 10205-10219, 2014 | 96 | 2014 |
Dietary gallic acid and anthocyanin cytotoxicity on human fibrosarcoma HT1080 cells. A study on the mode of action K Filipiak, M Hidalgo, JM Silvan, B Fabre, RJ Carbajo, A Pineda-Lucena, ... Food & function 5 (2), 381-389, 2014 | 41 | 2014 |
Progress towards water-soluble triazole-based selective MMP-2 inhibitors B Fabre, K Filipiak, JM Zapico, N Díaz, RJ Carbajo, AK Schott, ... Organic & Biomolecular Chemistry 11 (38), 6623-6641, 2013 | 40 | 2013 |
The development of a versatile trifunctional scaffold for biological applications V Vaněk, J Pícha, B Fabre, M Buděšínský, M Lepšík, J Jiráček European Journal of Organic Chemistry 2015 (17), 3689-3701, 2015 | 31 | 2015 |
Synthesis and evaluation of a library of trifunctional scaffold-derived compounds as modulators of the insulin receptor B Fabre, J Pícha, V Vaněk, I Selicharová, M Chrudinová, M Collinsová, ... ACS Combinatorial Science 18 (12), 710-722, 2016 | 30 | 2016 |
An integrated computational and experimental approach to gaining selectivity for MMP‐2 within the gelatinase subfamily B Fabre, K Filipiak, N Díaz, JM Zapico, D Suárez, A Ramos, ... ChemBioChem 15 (3), 399-412, 2014 | 27 | 2014 |
A CuAAC–hydrazone–CuAAC trifunctional scaffold for the solid-phase synthesis of trimodal compounds: possibilities and limitations B Fabre, J Pícha, V Vaněk, M Buděšínský, J Jiráček Molecules 20 (10), 19310-19329, 2015 | 21 | 2015 |
New clicked thiirane derivatives as gelatinase inhibitors: the relevance of the P1′ segment B Fabre, K Filipiak, C Coderch, JM Zapico, RJ Carbajo, AK Schott, ... RSC advances 4 (34), 17726-17735, 2014 | 12 | 2014 |
Tri‐Orthogonal Scaffolds for the Solid‐Phase Synthesis of Peptides J Pícha, B Fabre, M Buděšínský, J Hajduch, M Abdellaoui, J Jiráček European Journal of Organic Chemistry 2018 (37), 5180-5192, 2018 | 8 | 2018 |
Multipodal insulin mimetics built on adamantane or proline scaffolds J Hajduch, B Fabre, B Klopp, R Pohl, M Buděšínský, V Šolínová, ... Bioorganic chemistry 107, 104548, 2021 | 6 | 2021 |
ACS Comb. Sci., 2016, 18, 710;(d) A.-C. Knall, M. Hollauf, R. Saf and C. Slugovc B Fabre, J Pícha, V Vaněk, I Selicharová, M Chrudinová, M Collinsová, ... Org. Biomol. Chem 14, 10576, 2016 | 6 | 2016 |
Probing tripodal peptide scaffolds as insulin and IGF‐1 receptor ligands B Fabre, J Pícha, I Selicharová, L Žáková, M Chrudinová, J Hajduch, ... European Journal of Organic Chemistry 2018 (37), 5193-5201, 2018 | 3 | 2018 |
Targeting the insulin receptor with hormone and peptide dimers J Lin, I Selicharová, K Mitrová, B Fabre, VM Miriyala, M Lepšík, J Jiráček, ... Journal of Peptide Science 29 (4), e3461, 2023 | 1 | 2023 |
Combinatorial libraries of bipodal binders of the insulin receptor I Selicharová, B Fabre, M Soledad Garre Hernández, M Lubos, J Pícha, ... ChemMedChem 19 (11), e202400145, 2024 | | 2024 |
Progress towards water-soluble triazole-based selective MMP-2 inhibitors. A Ramos González, MP Martínez Alcázar, JM Zapico Rodríguez, ... | | 2013 |
Strategy to gain selectivity within the gelatinase subfamily. Design and synthesis of novel matrix metalloprotease-2 (mmp-2) inhibitors B Fabre Universidad CEU San Pablo, 2013 | | 2013 |