Current trends in computer aided drug design and a highlight of drugs discovered via computational techniques: A review VT Sabe, T Ntombela, LA Jhamba, GEM Maguire, T Govender, T Naicker, ... European Journal of Medicinal Chemistry 224, 113705, 2021 | 440 | 2021 |
Sulfonimidamides in medicinal and agricultural chemistry PK Chinthakindi, T Naicker, N Thota, T Govender, HG Kruger, ... Angewandte Chemie International Edition 56 (15), 4100-4109, 2017 | 182 | 2017 |
Asymmetric organocatalytic epoxidations: Reactions, scope, mechanisms, and applications RL Davis, J Stiller, T Naicker, H Jiang, KA Jørgensen Angewandte Chemie International Edition 53 (29), 7406-7426, 2014 | 145 | 2014 |
Beyond classical reactivity patterns: Shifting from 1, 4-to 1, 6-additions in regio-and enantioselective organocatalyzed vinylogous reactions of olefinic lactones with enals … L Dell’Amico, Ł Albrecht, T Naicker, PH Poulsen, KA Jørgensen Journal of the American Chemical Society 135 (21), 8063-8070, 2013 | 137 | 2013 |
Enantioselective organocatalyzed transformations of β-ketoesters T Govender, PI Arvidsson, GEM Maguire, HG Kruger, T Naicker Chemical Reviews 116 (16), 9375-9437, 2016 | 128 | 2016 |
Synthesis and biological evaluation of a teixobactin analogue YE Jad, GA Acosta, T Naicker, M Ramtahal, A El-Faham, T Govender, ... Organic letters 17 (24), 6182-6185, 2015 | 114 | 2015 |
A synthesis of “dual warhead” β-aryl ethenesulfonyl fluorides and one-pot reaction to β-sultams PK Chinthakindi, KB Govender, AS Kumar, HG Kruger, T Govender, ... Organic Letters 19 (3), 480-483, 2017 | 95 | 2017 |
NOTA: a potent metallo-β-lactamase inhibitor AM Somboro, D Tiwari, LA Bester, R Parboosing, L Chonco, HG Kruger, ... Journal of Antimicrobial Chemotherapy 70 (5), 1594-1596, 2015 | 80 | 2015 |
Organocatalytic asymmetric remote aziridination of 2, 4-dienals KS Halskov, T Naicker, ME Jensen, KA Jørgensen Chemical Communications 49 (57), 6382-6384, 2013 | 80 | 2013 |
On-water synthesis of biaryl sulfonyl fluorides PK Chinthakindi, HG Kruger, T Govender, T Naicker, PI Arvidsson The Journal of Organic Chemistry 81 (6), 2618-2623, 2016 | 56 | 2016 |
In vitro evaluation of metal chelators as potential metallo‐ β ‐lactamase inhibitors R Azumah, J Dutta, AM Somboro, M Ramtahal, L Chonco, R Parboosing, ... Journal of Applied Microbiology 120 (4), 860-867, 2016 | 51 | 2016 |
Re-evaluation of the N-terminal substitution and the D-residues of teixobactin SAH áAbdel Monaim, BG áde la Torre Rsc Advances 6 (77), 73827-73829, 2016 | 50 | 2016 |
N-Trifluoromethylthiolated Sulfonimidamides and Sulfoximines: Anti-microbial, Anti-mycobacterial, and Cytotoxic Activity N Thota, P Makam, KK Rajbongshi, S Nagiah, NS Abdul, AA Chuturgoon, ... ACS medicinal chemistry letters 10 (10), 1457-1461, 2019 | 43 | 2019 |
Novel tetrahydroisoquinoline based organocatalysts for asymmetric Diels–Alder reactions: insight into the catalytic mode using ROESY NMR and DFT studies T Naicker, K Petzold, T Singh, PI Arvidsson, HG Kruger, GEM Maguire, ... Tetrahedron: Asymmetry 21 (23), 2859-2867, 2010 | 37 | 2010 |
A 2018–2019 patent review of metallo beta-lactamase inhibitors N Reddy, M Shungube, PI Arvidsson, S Baijnath, HG Kruger, T Govender, ... Expert Opinion on Therapeutic Patents 30 (7), 541-555, 2020 | 35 | 2020 |
Sulfonimidamide in medizinischer Chemie und Agrochemie PK Chinthakindi, T Naicker, N Thota, T Govender, HG Kruger, ... Angewandte Chemie 129 (15), 4160-4170, 2017 | 34 | 2017 |
A new and facile access to the 2-(indol-3-yl)-3-nitriloquinolines based on Friedländer annulations M Shiri, MA Zolfigol, M Pirveysian, R Ayazi-Nasrabadi, HG Kruger, ... Tetrahedron 68 (30), 6059-6064, 2012 | 34 | 2012 |
Synthesis of tetrahydroisoquinoline-diamine ligands and their application in asymmetric transfer hydrogenation BK Peters, SK Chakka, T Naicker, GEM Maguire, HG Kruger, ... Tetrahedron: Asymmetry 21 (6), 679-687, 2010 | 33 | 2010 |
Asymmetric Organocatalytic Benzylation of α, β‐Unsaturated Aldehydes with Toluenes L Dell'Amico, X Companyó, T Naicker, TM Bräuer, KA Jørgensen European Journal of Organic Chemistry 2013 (24), 5262-5265, 2013 | 32 | 2013 |
Mass spectrometry imaging demonstrates the regional brain distribution patterns of three first-line antiretroviral drugs S Ntshangase, S Mdanda, SD Singh, T Naicker, HG Kruger, S Baijnath, ... ACS omega 4 (25), 21169-21177, 2019 | 31 | 2019 |